Top 5 Nootropics For Sleep

For me there is nothing I can’t stand more than not getting a good night's sleep.

Whether I can’t fall asleep or I just keep waking up all through the night is a real pain in the…well, you know.

Have you ever run into this problem?

What’s worse is the following day you feel like a zombie and have a hard time even getting the basics done.

The advice out there is also pretty worthless when it comes to helping out with this situation.

Stuff like “get more exercise” and “try to relax” really do no good for me.

So, what do I do when I can’t get to sleep?

I hack the problem with nootropics!

For this post I have got five nootropics that can help get you to sleep, keep you asleep, and boost the overall quality of your sleep.

Are ready to jump into in?

Cool, lets go…

Getting to sleep quickly

A lot of people out there have a hard time getting to sleep once they get in bed.

Has that ever happened to you?

 For the people out there who have problems falling asleep may be dealing with cognitive over-activity.

When this happens taking a nootropic that can inhibit neurotransmitters is going to turn down or turn off the excess stimulation that is going on up in your head.

So, here’s a super nootropic that you can use for getting to sleep quickly.

Nootropics for Sleep – Phenibut 

Phenibut Background Info

It was created back in the 1960’s by the Soviet Academy of Medical Sciences as drug to help treat anxiety and insomnia.

In the U.S. it has always been an over the counter supplement that has has been used to help with all kinds of issues that range from Anxiety to Stress and from Insomnia to PTSD.

Phenibut is a version of gamma-aminobutyric acid, GABA for short, but has been slightly modified.

By the way, GABA is naturally released by the brain to boost feelings of relaxation and calmness.

Phenibut not only helps to calm users down, but also helps out with things like anxiety, depression, fatigue, and stress.

But we’ll get to the benefits in a few minutes.

Now let’s jump right into how this stuff actually works.

How Phenibut Works

Like I mentioned above, Phenibut is a modified version of GABA but it has the ability to cross over the blood brain barrier to work its magic.

GABA is thought to be an inhibitor of excitatory action in the brain.

Basically it help balance out things like excessive brain activity that can happen when you are feeling over anxious.

What Phenibut does as soon as it gets up to the brain is stimulate GABA receptors on certain synaptic paths between neurons.

In case you are wondering Phenibut specifically it stimulates the GABA-A and GABA-B receptors.

Anyway, Phenibut also has plays a small part in stimulating dopamine receptors.

And as we all know dopamine plays a big part in boosting mood and feeling good.

In a really small nutshell that is how Phenibut works.

Now let’s keep moving and take a look at the benefits of this nootropic supplement.

Benefits of Phenibut

The biggest benefit of Phenibut is a its ability to reduce anxiety without slowing cognitive functions.

Other anxiolytics, like Xanax, for example tend to slow cognitive functions leaving you to process information much slower.

Basically you think and react slower.

Phenibut also helps out with improving your memory and boosting several cognitive processes.

Most important, for this post anyway, it is also a powerful sleep aid that not only helps you to get to sleep quickly, but helps with the quality of sleep so you feel more rested when you get out of bed.

Side Effects

Phenibut is known to be safe when it is used at low dosages.

When users go above the recommended dosage levels it can cause side effects close to the side effects related to benzodiazepines, GHB, and Alcohol.

The most common side effects of Phenibut are; fatigue, headache, stomach ache, nausea, and lightheadedness.

The more serious side effects include unconsciousness as well as memory loss.

People who use Phenibut constantly have been known to have withdrawal if they stop using it.

This is why if you plan on using it, using it only when you really need it is a good idea.

Lastly, always talk to a healthcare provider before you start using this or any other supplement of drug to ensure that it won’t cause any health issues for you.


Being that Phenibut is a strong drug, it is crazy important that you stay within the recommended guidelines.

The recommended dose is between 250 mg  and 1000 mg per day.

Just like most other strong nootropics it is a good idea to start off with small doses to see how your body is going to react and what side effects might pop up on you.

Phenibut has a long half life and the effects tend to last for quite some time, so it’s recommended to take it at least 4 hours apart if you decide to split up a daily dose into several parts.

Phenibut Stack Hack

Phenibut is great all by itself but some people like to get more out of, so the combine in with other supplements or nootropics which is known as stacking.

Stacking Phenibut with Aniracetam is a great way to get you brain calmed down and be totally relaxed with the dopamine targeting of the powerful Aniracetam.

This stack is perfect for when you need to get solid night’s sleep and wake up feeling totally refreshed.

Where to get it

If you head out to your local GNC or health food store you aren’t going to find Phenibut in the shelves.

But don’t worry,  you just have to hop online and do a quick google search for it.


You can check out

They have a big selection of nootropics, including Phenibut, that they can ship fast right to you.

One of the thing I really love about them is that they guarantee all there nootropics and supplements.

If you aren’t a 100% happy just send them back to and they’ll refund your money.

Just click the link below to head over to their site.

Click Here To Learn More About Phenibut

Staying Asleep

Another problem a lot of people run into during their sleep time is waking up over and over during the night.

Constantly waking up can cause real problems for not only your sleep cycle, but for your brain also.

You see, your brain need a break to for all the conscious actions it carries out during the day and needs time to work on repairing and making more cells for the brain.

Taking Phenibut right before you got to bed can help out a little here, but there is something better to use in my opinion.

So what nootropic supplements are going to help you stay asleep?

Let’s look at a two of them that can really help out.

Nootropics for Sleep – Aniracetam

Aniracetam Background Info

Aniracetam was created in 1970 as an analog to the original nootropic Piracetam.

The Belgian pharma company Hoffmann-La Roche developed it to boost brain function and aid in treatment of cognitive problems.

Throughout much of Western Europe it is still prescribed as a treatment for cognitive issues and sleep disorders.

In the United States it is sold as a nootropic supplement that does not require a prescription.

How it works

Aniracetam primarily works by boosting two neurotransmitters that make us feel really good.

Those two are Dopamine and Serotonin.

They play a big part when it comes to boosting mood and keeping us relaxed.

Aniracetam also starts to boost AMPA receptor sites and what is awesome about these sites is that they speed up synaptic communication in the nervous system.

At its most basic level Aniracetam boosts neural communication and cranks up dopamine and serotonin to keep us chilled out.


Like Phenibut, the major benefit of Aniracetam is a boost in mood.

Aniracetam targets two of the  dopamine and serotonin receptors that help to lower levels of depression, stress, and provide an overall relaxed sense.

Like I already mentioned, when your body is relaxed it's going to help give you a much better quality of sleep.

In addition to a boost in overall mood, Aniracetam also boosts mental energy, gives users clarity of thought and has a noticeable effect on memory.

Side effects

Aniracetam is considered to be safe and has a low toxicity to the body, but does has some side effects.

Side effects tend to happen when you get into the higher end of the dosage scale.

Headaches,nausea, insomnia, and GI tract distress are the most common side effects that you are likely to run into if you run to any at all.


Aniracetam is commonly dosed at 750 mg twice daily is either powder or capsule form.

It is recommended that if you are new to using Aniracetam that you start off with a smaller than normal dose.

350 mg to 400 mg is a good place to start for new users.

This is so you will have an idea of the effects on your brain and if any of the side effects pop up.

Lastly, Aniracetam is fat soluble so it is a good idea to take with something like fish oil or even milk.

Stack Hack

Stacking Aniracetam and Alpha GPC together is a solid way to avoid side effects and boost dream states.

As we just went over Aniracetam is great for getting you relaxed and ready for restful deep sleep.

But when it’s stacked with  Alpha GPC you’ll reduce or get rid of headaches that tend to happen when taking Aniracetam and is a powerful way to induce lucid dreaming.

Where to get it

Just like with Phenibut, you are going to most likely to order Aniracetam online because it’s not going to be sold at the local GNC.

Heck, it’s not even sold on

But, has got it. Plus they have a bunch of other nootropics and supplements you can check out.

I’ve been getting just about all my nootropics from them for quite a while now and I couldn't be happier.

Only once have I ever had a problem and that turned out to be a good thing.

That’s right, a problem turned into a good thing!

That just another of the many reasons that I continue to order stuff like Aniracetam  from the team at

Click Here to Learn More About Aniracetam

Nootropics for Sleep – Picamilon

Picamilon Background Info

In 1969 at the Soviet Scientific Research Institute for Vitamins scientists created Picamilon for treating depression, migraines, and different forms of glaucoma.

At its most basic Picamilon is a combination of GABA and Naicin joined together to help GABA get across the blood brain barrier.

It is still used widely in Eastern Europe as a prescription drug for treating different types of sleep related issues.

In the western world it is used mostly to help lower stress and anxiety and is sold as an over the counter supplement.

How it works

Picamilon gets across the blood brain barrier by way of Naicin pathway to the brain and is then broken down into GABA and Naicin.

At this point the good stuff starts to happen.

The broken down Picamilon provides the brain with higher amounts of GABA which I mentioned above is a inhibiting neurotransmitter.

Basically your brain becomes balanced out and calm from the over excitement of over active synaptic transmission.

You know, you have lower stress, anxiety and are able to really relax.

Benefits of Picamilon

The most prominent benefits of this nootropic are a boost in mood and improvement in brain function.

What most users tend to get when taking Picamilon is a lower levels of stress and anxiety as well as a positive outlook and attitude.

When we are relaxed we tend to get a better and more restful night’s sleep.

And that’s just something we could all use more of.

Anyway, Picamilon also helps boost mental energy and mental clarity.

Some users take it on a regular basis to simply help them relax and some people use it to make it easier to think.

Either way, you’ll be relaxed and it is going to help you get to sleep quickly.

Side effects

The side effects of Picamilon are very mild and rarely occurring and there has never been any published reports of serious side effects.

Common side effects include;headaches, fatigue, and GI discomfort, and nervousness.

For the majority of users that run into side effects is simply caused by taking way too much of this supplement.

By cutting down on dosage is what is recommended to help cut out side effects from Picamilon.


Most makers of Picamilon recommend that users take between 50mg and 100mg daily.

With that being said, many users take between 100mg and 200mg a day for better anxiety and stress relief.

It is safe for daily use, but a lot of people cycle it to avoid building up a tolerance.

Even though Picamilon is considered safe for daily use it is best you speak with a doctor or healthcare provider to find out what the best dose for your situation is best.

Picamilon Stack Hack

L-Theanine and Picamilon make a super combo for solid sleep

The L-Theanine boost alpha waves in the brain that brings on a calming effect and boosts deep sleep while the Picamilon lowers anxiety that in turn boosts relaxation for better sleep.

Where to get it

Very few stores in the North American Market are going to carry Picamilon, so getting it online is going to be the easiest way to pick some up.

I have ordered Picamilon from once before, but I didn’t think it was the best quality so I found another decent place to get it.

I ordered it from Serious Nutrition

Unfortunately doesn’t sell Picamilon, but they do have a ton of different nootropics you can check out.

Quality sleep

So let’s say you can get to sleep and stay knocked out all night, how many time have you woken up after six or seven hours feeling like you only slept a few minutes?

It’s happened to me more times than I can count.

Waking up in foggy and unfocused way totally sucks.

A lot of times you get the “foggy” feeling because you were woken up during a REM cycle of sleep.

Sometimes this feeling comes from not getting enough deep sleep during the night.

Without getting to some deep neuroscience here, there 5 stages of sleep that your body and brain go through during sleep.

Stage 1 and 2 are basic sleep, but not a deep sleep.

Stage 3 and 4 are deep sleep where you breathing and heartrate have slowed down.

Stage 5 is the REM (rapid eye movement) stage. Your eyes are moving around and the brain is crazy active. This is the stage where you are dreaming

Normally we go through 5 or 6 of these complete cycles during the night.  

With all that being said there are a couple of super nootropics that can boost the deep sleep cycle and help out with getting more powerful sleep during the REM cycle.

Nootropics for Sleep – L-Theanine

Background info

Gamma-glutamylethylamide, commonly known as L-Theanine, is the analog of glutamate and glutamine that is able to boost and modulate alpha brain waves in the brain.

In 1949 L-Theanine was discovered in green tea and the major component was soon extracted for testing and research.

The nootropic benefits of L-Theanine weren't really discovered until 1999 when the Food Science and Technology Research Institute found that weekly doses could boost cognitive function.

Today it is commonly sold as an over counter supplement throughout most of the western world.

How it works

The specifics of how L-Theanine works are not completely known, but it is able to cross over the blood brain barrier and it gets to work really fast.

Once it get into the brain it targets Serotonin, Dopamine, GABA, as well as Norpinephrine.

These neurotransmitters play a big part in cognitive areas, the pleasure and reward system of the brain and most importantly for this article sleep and relaxation cycles.


The main benefits of L-theanine affect your mood, general health and cognitive functions.

What most people tend to get is a relaxed and peaceful feeling along with a optimistic outlook on things in general.

L-Theanine also boosts Alpha waves in the brain.

These waves produce mental alertness and clarity while feeling very calm.

Lastly, it has also been seen to have an antioxidant effect on LDL cholesterol and know to help reduce blood pressure by opening blood vessels in the arteries.

Side effects and Interactions

One of the great things of L-Theanine is that there are no known side effects.

With that being said, large doses of this supplement have been reportedly known to cause some diarrhea in some people.

You should avoid using L-Theanine with stimulants because their effects will be dramatically decreased.

Lastly, avoid using it with meds that are for treating high blood pressure.

The combination may lower blood pressure to dangerously low levels.


The minimum dose for positive effects of L-Theanine is 50mg.

It’s basically a starter dose.

Try taking it all by itself without other supplement and pay attention to how you feel

Slowly increase the the dosage by 50mg and see how it goes.

Most users take the median dose of around 200 mg to 250 mg per day.

It is recommended that you cap your dose at no more than 400mg per day.

L-Theanine Stack Hack

Are you looking for some incredible restful deep sleep?

Stacking a Aniracetam on top of L-Theanine is going give you just that.

As the L-Theanine boosts Alpha waves in the brain and its calming kick in the Aniracetam begins to target the dopamine and serotonin receptors to relax your body for sleep.

Where to get it

L-Theanine is a supplement that you shouldn’t have a problem getting a hold of.

From GNC to Wal-Mart or anywhere with a vitamin and supplement section is probably going to have this stuff.

Even though you can get it about anywhere, I would suggest you get the best quality L-Theanine you can.

So, where do you get the best and highest quality L-Theanine?

That's easy…

So why order from them?

Also, really easy.

Not only do they they have super customer service, a money back guarantee, but they also have all their nootropics tested by a third party lab to ensure at least 98% purity.

So for me, it's a no brainier to order from them.

Click Here To Learn More About L-Theanine

Nootropics for Sleep – Huperzine-A

Background Info

Huperzine comes from the Chinese moss Huperzia Serrata and is classed as an alkaloid.

For the most part is is used as a cognitive booster and memory enhancer.

Interestingly enough, it also works to boost neuroplasticity in the brain.

That’s the forming of new neural pathways and synapses that help people learn faster and remember more.

How it works

Huperzine-A work a lot like some members of the racetam family on the cholinergic system in your brain.

But instead of boosting acetylcholine receptors, like Piracetam for example, it inhibits an enzyme that breaks down acetylcholine from being used again by the neurons in your brain.

Because Huperzine-A blocks Acetylcholinesterase from breaking down acetylcholine there is more of the acetylcholine to boost memory, focus, learning, and reasoning ability.

Without all the science talk, basically Huperzine-A boosts the neurons in your brain to be able to connect with each other.


The primary benefit of Huperzine-A gives your memory a real boost as well help out with learning.

But when it come to using the bad ass nootropic for sleep it can boost REM sleep cycles by as much as 30%.

Side effects

First off, Huperzine-A is known to be very safe and has no toxicity to the body when taken in the recommended dosages.

The most common side effects include, nausea, vomiting and diarrhea.

Other side effects that happen rarely include, increased salivation, restlessness, blurred vision, and slurred speech.

These side effects, just in case you run into them, are not life threatening or long term.

If you are taking any medications or suffering from any medical condition it is important that you talk with your healthcare provider to make sure that taking Huperzine-A is not going to cause any other complications.


Huperzine-A is a really concentrated drug that is taken in micro grams.

That’s 1/1000 of a milligram.

So yeah, that’s a really small number, but anyway…

Recommended daily dosages range from between 100 mcg to 200 mcg.

As with most nootropics, it is a good idea to start with small doses to see how you body and brain react.

To get the most out of Huperzine-A it is a good idea to stack with a member of the racetam family and/or a choline supplement.

When it comes to using this supplement as a sleep aid it is best to take it roughly 30 minutes prior to sleep.

Stack Hack

Huperzine-A Stacked with Aniracetam.

Like I mentioned above, stacking Huperzine-A with a racetam is a good idea to get the most out of Huperzine-A.

Stacking Huperzine-A is going to boost the REM cycles of sleep which is going to make you feel like you had super quality sleep.

Aniracetam is going to get your body relaxed to help you get to sleep easier.

Where to get it

Huperzine-A is for sure easy to find, just not as easy as L-Theanine.

You can get it GNC and some health food stores and tons of places online.

Got any info to share about nootropics and sleep? Share with everybody down in the comments section below!

3 thoughts on “Top 5 Nootropics For Sleep”

  1. Wonderful article!!!! It’s hard to find good enough like this all in one article. Would love to have you on my podcast if you would be interested? If so feel free to email me back!

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